5-Bromo-1,2-benzisoxazol-3-ylamine

• CAS: 455280-00-9
• Catalog Number: ACM455280009
• Category: Other Products
• Molecular Formula: C₇H₅BrN₂O
• Synonyms: 5-Bromo-1,2-benzisoxazol-3-ylamine;5-Bromobenzo[d]isoxazol-3-ylamine

Synthetic Use

Upstream Synthesis Route 1

• 546-88-3
• 179897-89-3

• 455280-00-9

Reference: [1] Patent: WO2010/138488, 2010, A1, . Location in patent: Page/Page column 57-58

Upstream Synthesis Route 2

• 179897-89-3

• 455280-00-9

Reference: [1] Journal of Medicinal Chemistry, 2014, vol. 57, # 18, p. 7624 - 7643
[2] Patent: WO2006/122799, 2006, A1, . Location in patent: Page/Page column 60-61
[3] ACS Medicinal Chemistry Letters, 2016, vol. 7, # 3, p. 277 - 282

Upstream Synthesis Route 3

• 179897-89-3

• 455280-00-9

Reference: [1]Patent: WO2019/108943,2019,A1 .Location in patent: Paragraph 0280; 0352-0354

Upstream Synthesis Route 4

• 546-88-3
• 179897-89-3

• 455280-00-9

Reference: [1]Patent: WO2019/243491,2019,A1 .Location in patent: Page/Page column 83

Downstream Synthesis Route 1

• 455280-00-9
• 75-36-5

• 1404480-08-5

Reference: [1]Patent: WO2010/51042,2010,A1 .Location in patent: Page/Page column 134

* For details of the synthesis route, please refer to the original source to ensure accuracy.